A new route to iodine-labeled N-isopropyl iodoamphetamine via organoboranes

George Kabalka, Rajender S. Varma, Yuan Zhu Gai, Ronald M. Baldwin

Research output: Contribution to journalArticle

16 Citations (Scopus)

Abstract

N-Isopropyl amphetamineboronic acid was prepared via a new in-situ transmetallation reaction involving sonication. The boronic acid intermediate was radioiodinated via a novel iodination procedure.

Original languageEnglish (US)
Pages (from-to)3843-3844
Number of pages2
JournalTetrahedron Letters
Volume27
Issue number33
DOIs
StatePublished - Jan 1 1986
Externally publishedYes

Fingerprint

Boronic Acids
Sonication
Halogenation
Iodine
Acids

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Drug Discovery
  • Organic Chemistry

Cite this

A new route to iodine-labeled N-isopropyl iodoamphetamine via organoboranes. / Kabalka, George; Varma, Rajender S.; Gai, Yuan Zhu; Baldwin, Ronald M.

In: Tetrahedron Letters, Vol. 27, No. 33, 01.01.1986, p. 3843-3844.

Research output: Contribution to journalArticle

Kabalka, George ; Varma, Rajender S. ; Gai, Yuan Zhu ; Baldwin, Ronald M. / A new route to iodine-labeled N-isopropyl iodoamphetamine via organoboranes. In: Tetrahedron Letters. 1986 ; Vol. 27, No. 33. pp. 3843-3844.
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