Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Vipin A. Nair, Suni M. Mustafa, Michael L. Mohler, Jun Yang, Leonid I. Kirkovsky, James T. Dalton, Duane Miller

Research output: Contribution to journalArticle

11 Citations (Scopus)

Abstract

A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.

Original languageEnglish (US)
Pages (from-to)4821-4823
Number of pages3
JournalTetrahedron Letters
Volume46
Issue number28
DOIs
StatePublished - Jul 11 2005

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Androgen Receptors
Ligands
Imaging techniques
bicalutamide

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Drug Discovery
  • Organic Chemistry

Cite this

Nair, V. A., Mustafa, S. M., Mohler, M. L., Yang, J., Kirkovsky, L. I., Dalton, J. T., & Miller, D. (2005). Synthesis of irreversibly binding bicalutamide analogs for imaging studies. Tetrahedron Letters, 46(28), 4821-4823. https://doi.org/10.1016/j.tetlet.2005.04.143

Synthesis of irreversibly binding bicalutamide analogs for imaging studies. / Nair, Vipin A.; Mustafa, Suni M.; Mohler, Michael L.; Yang, Jun; Kirkovsky, Leonid I.; Dalton, James T.; Miller, Duane.

In: Tetrahedron Letters, Vol. 46, No. 28, 11.07.2005, p. 4821-4823.

Research output: Contribution to journalArticle

Nair, VA, Mustafa, SM, Mohler, ML, Yang, J, Kirkovsky, LI, Dalton, JT & Miller, D 2005, 'Synthesis of irreversibly binding bicalutamide analogs for imaging studies', Tetrahedron Letters, vol. 46, no. 28, pp. 4821-4823. https://doi.org/10.1016/j.tetlet.2005.04.143
Nair VA, Mustafa SM, Mohler ML, Yang J, Kirkovsky LI, Dalton JT et al. Synthesis of irreversibly binding bicalutamide analogs for imaging studies. Tetrahedron Letters. 2005 Jul 11;46(28):4821-4823. https://doi.org/10.1016/j.tetlet.2005.04.143
Nair, Vipin A. ; Mustafa, Suni M. ; Mohler, Michael L. ; Yang, Jun ; Kirkovsky, Leonid I. ; Dalton, James T. ; Miller, Duane. / Synthesis of irreversibly binding bicalutamide analogs for imaging studies. In: Tetrahedron Letters. 2005 ; Vol. 46, No. 28. pp. 4821-4823.
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