Synthesis of novel iodo derived bicalutamide analogs

Vipin A. Nair, Suni M. Mustafa, Michael L. Mohler, Scott J. Fisher, James T. Dalton, Duane Miller

Research output: Contribution to journalArticle

20 Citations (Scopus)

Abstract

A series of optically active nonsteroidal selective androgen receptor modulators with structures analogous to bicalutamide was prepared by replacing the trifluoromethyl group with iodine and the sulfonyl linker by oxygen.

Original languageEnglish (US)
Pages (from-to)9475-9477
Number of pages3
JournalTetrahedron Letters
Volume45
Issue number51
DOIs
StatePublished - Dec 13 2004
Externally publishedYes

Fingerprint

Androgen Receptors
Iodine
Modulators
Oxygen
bicalutamide

All Science Journal Classification (ASJC) codes

  • Biochemistry
  • Organic Chemistry
  • Drug Discovery

Cite this

Nair, V. A., Mustafa, S. M., Mohler, M. L., Fisher, S. J., Dalton, J. T., & Miller, D. (2004). Synthesis of novel iodo derived bicalutamide analogs. Tetrahedron Letters, 45(51), 9475-9477. https://doi.org/10.1016/j.tetlet.2004.10.130

Synthesis of novel iodo derived bicalutamide analogs. / Nair, Vipin A.; Mustafa, Suni M.; Mohler, Michael L.; Fisher, Scott J.; Dalton, James T.; Miller, Duane.

In: Tetrahedron Letters, Vol. 45, No. 51, 13.12.2004, p. 9475-9477.

Research output: Contribution to journalArticle

Nair, VA, Mustafa, SM, Mohler, ML, Fisher, SJ, Dalton, JT & Miller, D 2004, 'Synthesis of novel iodo derived bicalutamide analogs', Tetrahedron Letters, vol. 45, no. 51, pp. 9475-9477. https://doi.org/10.1016/j.tetlet.2004.10.130
Nair VA, Mustafa SM, Mohler ML, Fisher SJ, Dalton JT, Miller D. Synthesis of novel iodo derived bicalutamide analogs. Tetrahedron Letters. 2004 Dec 13;45(51):9475-9477. https://doi.org/10.1016/j.tetlet.2004.10.130
Nair, Vipin A. ; Mustafa, Suni M. ; Mohler, Michael L. ; Fisher, Scott J. ; Dalton, James T. ; Miller, Duane. / Synthesis of novel iodo derived bicalutamide analogs. In: Tetrahedron Letters. 2004 ; Vol. 45, No. 51. pp. 9475-9477.
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